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Found 4 Enz. Inhib. hit(s) with Target = 'Methionine aminopeptidase' and Ligand = 'BDBM50129661'
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129661(CHEMBL89671 | N-(thiazol-2-yl)picolinamide | Pyrid...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibitory concentration against Escherichia coli methionine aminopeptidase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129661(CHEMBL89671 | N-(thiazol-2-yl)picolinamide | Pyrid...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibitory activity against Methionine aminopeptidase 1 from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129661(CHEMBL89671 | N-(thiazol-2-yl)picolinamide | Pyrid...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibitory concentration required against Escherichia coli MetAP1 (150 nM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50129661(CHEMBL89671 | N-(thiazol-2-yl)picolinamide | Pyrid...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibitory concentration against EcMetAP1 enzyme activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed