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Found 3 Enz. Inhib. hit(s) with Target = 'Mu-type opioid receptor' and Ligand = 'BDBM50252861'
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50252861(CHEMBL507214 | H-D-Phe-c[Cys-Tyr-DTrp-Orn-Thr-Pen]...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]DAMGO from MOR in rat brain membrane measured after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50252861(CHEMBL507214 | H-D-Phe-c[Cys-Tyr-DTrp-Orn-Thr-Pen]...)
Affinity DataIC50:  2.80nMAssay Description:Compound was evaluated for the inhibition of binding of [3H]naloxone toOpioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50252861(CHEMBL507214 | H-D-Phe-c[Cys-Tyr-DTrp-Orn-Thr-Pen]...)
Affinity DataIC50:  2.80nMAssay Description:Antagonist activity against mu opioid receptor in guinea pig ileum assessed as effect on TAPP-induced responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed