Affinity DataKi: 69nMAssay Description:Displacement of [3H]DAMGO from mu-opioid receptor in Sprague-Dawley rat brain membrane after 180 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 148nMAssay Description:Displacement of [3H]DAMGO from mu-opioid receptor in Sprague-Dawley rat brain membrane after 180 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.01E+3nMAssay Description:Agonist activity at mu-opioid receptor in Hartley guinea pig isolated ileum assessed as inhibition of contraction in electrically stimulated muscleMore data for this Ligand-Target Pair