Found 2 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1' and Ligand = 'BDBM50038707'
Affinity DataKi: 880nMAssay Description:Binding affinity was measured as selectivity for sigma-1 site over muscarinic (M1) receptor in rat using [3H]pirenzepine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >1.76E+4nMAssay Description:The nitro derivative RLH-033 shows significant selectivity for the [3H]-(=)-PENT site over muscarinic 1 in rat using [3H]pirenzepine as radioligandMore data for this Ligand-Target Pair