Compile Data Set for Download or QSAR
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Found 1 Enz. Inhib. hit(s) with Target = 'NAD-dependent protein deacetylase sirtuin-1' and Ligand = 'BDBM50358043'
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Ludwig-Maximilians-Universit£T M£Nchen

Curated by ChEMBL
LigandPNGBDBM50358043(CHEMBL1794051 | GW-5074)
Affinity DataIC50:  4.16E+4nMAssay Description:Inhibition of human recombinant N-terminally GST-tagged SIRT1 after 4 hrs in presence of NAD+ by fluorescent deacetyalse assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed