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Found 4 Enz. Inhib. hit(s) with Target = 'NAD-dependent protein deacylase sirtuin-5, mitochondrial' and Ligand = 'BDBM50540057'
TargetNAD-dependent protein deacylase sirtuin-5, mitochondrial(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50540057(CHEMBL4636862)
Affinity DataKi:  6nMAssay Description:Binding affinity to SIRT5 (unknown origin) assessed as deglutarylase activity by measuring inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNAD-dependent protein deacylase sirtuin-5, mitochondrial(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50540057(CHEMBL4636862)
Affinity DataIC50:  110nMAssay Description:Inhibition of SIRT5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-5, mitochondrial(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50540057(CHEMBL4636862)
Affinity DataIC50:  110nMAssay Description:Inhibition of SIRT5 deglutarylase activity (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNAD-dependent protein deacylase sirtuin-5, mitochondrial(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50540057(CHEMBL4636862)
Affinity DataIC50: <300nMAssay Description:Inhibition of SIRT5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed