Affinity DataKi: 4.60nMAssay Description:Displacement of [125I][Tyr14]nociceptin/orphanin FQ from human nociceptin opioid receptor expressed in CHO cell membranes after 1 hr by microplate sc...More data for this Ligand-Target Pair
Affinity DataEC50: 79nMAssay Description:Agonist activity at human nociceptin opioid receptor expressed in CHO cell membranes after 30 mins by GTPgamma(35)S binding assayMore data for this Ligand-Target Pair