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Found 3 Enz. Inhib. hit(s) with Target = 'Nuclear receptor ROR-gamma' and Ligand = 'BDBM50044251'
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Innov17

US Patent
LigandPNGBDBM50044251(CHEMBL3314037 | US9321750, 2)
Affinity DataIC50: <1.00E+4nMAssay Description:Compound binding to the human RORγ LBD was assessed using the Human RORγ Assay System (INDIGO Biosciences Inc.) as per manufacturer's i...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Innov17

US Patent
LigandPNGBDBM50044251(CHEMBL3314037 | US9321750, 2)
Affinity DataEC50: <1.00E+4nMAssay Description:Inverse agonist activity at human RoRc in human skin model assessed as suppression of IL-17A level relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Innov17

US Patent
LigandPNGBDBM50044251(CHEMBL3314037 | US9321750, 2)
Affinity DataEC50: <1.00E+4nMAssay Description:Inverse agonist activity at human RoRc in human skin model assessed as suppression of IL-17F level relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed