Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Nuclear receptor ROR-gamma' and Ligand = 'BDBM50067722'
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50067722(CHEMBL3402135)
Affinity DataIC50:  2.20E+3nMAssay Description:Inverse agonist activity at RORC ligand binding domain (unknown origin) expressed in HEK293 cells transfected with GAL4 promoter by luciferase report...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50067722(CHEMBL3402135)
Affinity DataKd:  2.40E+3nMAssay Description:Binding affinity to RORC-SRC2 fusion construct (unknown origin) by TAMRA-labeled active site probe based fluorescence polarization competition bindin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed