Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Oxysterols receptor LXR-beta' and Ligand = 'BDBM50184273'
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50184273(2-(5-(methyl(3-(7-propyl-3-(trifluoromethyl)benzo[...)
Affinity DataIC50:  40nMAssay Description:Inhibition of LXR betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50184273(2-(5-(methyl(3-(7-propyl-3-(trifluoromethyl)benzo[...)
Affinity DataEC50:  150nMAssay Description:Activity at LXR beta as beta-lactamase transactivation in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed