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Found 12 Enz. Inhib. hit(s) with Target = 'P2X purinoceptor 4' and Ligand = 'BDBM50506159'
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer

Curated by ChEMBL
LigandPNGBDBM50506159(CHEMBL1532400)
Affinity DataIC50:  500nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in human HEK293 cells at -60 mv holding potential by Whole cell patch-clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer

Curated by ChEMBL
LigandPNGBDBM50506159(CHEMBL1532400)
Affinity DataIC50:  540nMAssay Description:Antagonist activity at human P2X4R transfected in HEK293 cells assessed as inhibition of ATP-evoked current by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer

Curated by ChEMBL
LigandPNGBDBM50506159(CHEMBL1532400)
Affinity DataIC50:  540nMAssay Description:Antagonist activity at human P2X4R transfected in HEK293 cells assessed as inhibition of ATP-evoked current by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer

Curated by ChEMBL
LigandPNGBDBM50506159(CHEMBL1532400)
Affinity DataIC50:  550nMAssay Description:Antagonist activity at human P2X4R transfected in 1321N1 cells assessed as inhibition of ATP-mediated calcium influx measured after 10 mins by Fura-2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer

Curated by ChEMBL
LigandPNGBDBM50506159(CHEMBL1532400)
Affinity DataIC50:  550nMAssay Description:Antagonist activity at human P2X4R transfected in 1321N1 cells assessed as inhibition of ATP-mediated calcium influx measured after 10 mins by Fura-2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer

Curated by ChEMBL
LigandPNGBDBM50506159(CHEMBL1532400)
Affinity DataIC50:  780nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in human HEK293 cells assessed as inhibition of ATP-induced calcium influx by Fluo2-AM staining...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer

Curated by ChEMBL
LigandPNGBDBM50506159(CHEMBL1532400)
Affinity DataIC50:  904nMAssay Description:Antagonist activity against human P2X4R stably transfected in human 1321N1 cells incubated for 30 mins by Fura-2 AM staining based calcium influx ass...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer

Curated by ChEMBL
LigandPNGBDBM50506159(CHEMBL1532400)
Affinity DataIC50:  1.30E+3nMAssay Description:Antagonist activity at human P2X4R transfected in HEK293 cells assessed as inhibition of ATP-mediated calcium influx measured after 10 mins by YOPRO-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer

Curated by ChEMBL
LigandPNGBDBM50506159(CHEMBL1532400)
Affinity DataIC50:  1.30E+3nMAssay Description:Antagonist activity at human P2X4R transfected in HEK293 cells assessed as inhibition of ATP-mediated calcium influx measured after 10 mins by YOPRO-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer

Curated by ChEMBL
LigandPNGBDBM50506159(CHEMBL1532400)
Affinity DataIC50:  1.60E+3nMAssay Description:Antagonist activity at human P2X4R transfected in 1321N1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer

Curated by ChEMBL
LigandPNGBDBM50506159(CHEMBL1532400)
Affinity DataIC50:  1.60E+3nMAssay Description:Antagonist activity at human P2X4R transfected in 1321N1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer

Curated by ChEMBL
LigandPNGBDBM50506159(CHEMBL1532400)
Affinity DataIC50:  1.95E+3nMAssay Description:Antagonist activity at P2X4R (unknown origin) expressed in 1321N1 cellsMore data for this Ligand-Target Pair
In DepthDetails PubMed