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Found 1 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor alpha' and Ligand = 'BDBM33289'
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Pfizer

LigandPNGBDBM33289(phenylpropanoic acid derivative, 17e)
Affinity DataIC50:  899nM EC50:  874nMpH: 7.2 T: 2°CAssay Description:Human PPAR alpha receptor was expressed as recombinant glutathione-S-transferase (GST)-fusion proteins in Escherichia coli. The purified GST-hPPAR al...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed