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Found 3 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor delta' and Ligand = 'BDBM323597'
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Mitobridge

US Patent
LigandPNGBDBM323597((E)-6-(2-((4-(furan-2-yl)-N-methylbenzamido)methyl...)
Affinity DataEC50:  694nMAssay Description:Medium including test compound was aspirated and washed with PBS. 50 μl PBS including 1 mM Mg++ and Ca++ were then added to each well. The lucif...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Mitobridge

US Patent
LigandPNGBDBM323597((E)-6-(2-((4-(furan-2-yl)-N-methylbenzamido)methyl...)
Affinity DataEC50:  690nMAssay Description:Activation of human PPARdelta LBD expressed in CHO-K1 cells by beta galactosidase enzyme fragment complement based fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Mitobridge

US Patent
LigandPNGBDBM323597((E)-6-(2-((4-(furan-2-yl)-N-methylbenzamido)methyl...)
Affinity DataEC50: >1.00E+4nMAssay Description:Transactivation of yeast GAL4 DNA binding domain-fused PPARdelta LBD (unknown origin) expressed in CV-1 cells after 24 hrs by luciferase reporter gen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed