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Found 2 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor gamma' and Ligand = 'BDBM50362958'
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362958(CHEMBL1946758)
Affinity DataIC50:  4.10nMAssay Description:Binding affinity to human PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50362958(CHEMBL1946758)
Affinity DataEC50:  13.2nMAssay Description:Agonist activity at human PPARgamma expressed in COS-1 cells co-expressing with Gal4 by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed