Found 1 Enz. Inhib. hit(s) with Target = 'Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform' and Ligand = 'BDBM50543091'
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Affinity DataIC50: 4.30nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using PIP2:3PS peptide as substrate preincubated for 15 mins followed by ATP addition at Km concentration an...More data for this Ligand-Target Pair