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Found 4 Enz. Inhib. hit(s) with Target = 'Poly [ADP-ribose] polymerase 1' and Ligand = 'BDBM50297828'
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Central South University

Curated by ChEMBL
LigandPNGBDBM50297828(7-(piperidin-1-ylmethyl)pyrrolo[1,2-a]quinoxalin-4...)
Affinity DataKi:  9nMAssay Description:Inhibition of PARP-1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Central South University

Curated by ChEMBL
LigandPNGBDBM50297828(7-(piperidin-1-ylmethyl)pyrrolo[1,2-a]quinoxalin-4...)
Affinity DataKi:  9nMAssay Description:Inhibition of PARP1 by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Central South University

Curated by ChEMBL
LigandPNGBDBM50297828(7-(piperidin-1-ylmethyl)pyrrolo[1,2-a]quinoxalin-4...)
Affinity DataEC50:  11nMAssay Description:Inhibition of PARP-1 (unknown origin) in cellular based assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Central South University

Curated by ChEMBL
LigandPNGBDBM50297828(7-(piperidin-1-ylmethyl)pyrrolo[1,2-a]quinoxalin-4...)
Affinity DataEC50:  11nMAssay Description:Inhibition of PARP1 in human C41 cells by DAPI staining-based FITC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed