Found 4 Enz. Inhib. hit(s) with Target = 'Proteasome subunit beta type-1' and Ligand = 'BDBM50444909' TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataKi: 340nMAssay Description:Competitive inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate Linewea...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 430nMAssay Description:Inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate measured for 1 hr b...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 720nMAssay Description:Inhibition of PGPH activity of human 20S proteasome using Z-LLE-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of PGPH activity of human 26S proteasome using Z-LLE-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
