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Found 2 Enz. Inhib. hit(s) with Target = 'Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha' and Ligand = 'BDBM50298242'
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50298242((E)-4-(3-benzoylbenzyloxy)-3-methylbut-2-enyl diph...)
Affinity DataKi:  610nMAssay Description:Inhibition of Saccharomyces cerevisiae protein farnesyltransferase assessed as farnsylation of N-dansyl-GCVIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50298242((E)-4-(3-benzoylbenzyloxy)-3-methylbut-2-enyl diph...)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of Saccharomyces cerevisiae protein farnesyltransferase assessed as farnsylation of N-dansyl-GCVIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed