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Found 2 Enz. Inhib. hit(s) with Target = 'Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha' and Ligand = 'BDBM50298245'
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50298245(4-Benzoylbenzylphosphonic((2E,6E)-3,7,11-trimethyl...)
Affinity DataKi:  480nMAssay Description:Inhibition of Saccharomyces cerevisiae protein farnesyltransferase assessed as farnsylation of N-dansyl-GCVIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50298245(4-Benzoylbenzylphosphonic((2E,6E)-3,7,11-trimethyl...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of Saccharomyces cerevisiae protein farnesyltransferase assessed as farnsylation of N-dansyl-GCVIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed