Found 3 Enz. Inhib. hit(s) with Target = 'Protein-glutamine gamma-glutamyltransferase 2' and Ligand = 'BDBM185181'
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
University Of Ottawa
Curated by ChEMBL
University Of Ottawa
Curated by ChEMBL
Affinity DataKi: 1.31E+3nMAssay Description:Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assayMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
University Of Ottawa
Curated by ChEMBL
University Of Ottawa
Curated by ChEMBL
Affinity DataKi: 1.49E+3nMAssay Description:Inhibition of recombinant human TG2 expressed in Escherichia coli assessed as inhibition constant using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) a...More data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
University Of Ottawa
Curated by ChEMBL
University Of Ottawa
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of recombinant human TG2 by fluorescence assayMore data for this Ligand-Target Pair