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Found 2 Enz. Inhib. hit(s) with Target = 'Proteinase-activated receptor 1' and Ligand = 'BDBM50079756'
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Oregon Health & Science University

Curated by ChEMBL
LigandPNGBDBM50079756(7-(4-Isopropyl-benzyl)-7H-pyrrolo[3,2-f]quinazolin...)
Affinity DataIC50:  300nMAssay Description:Antagonist activity at PAR1 (unknown origin) assessed as inhibition of thrombin-induced platelet aggregationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Oregon Health & Science University

Curated by ChEMBL
LigandPNGBDBM50079756(7-(4-Isopropyl-benzyl)-7H-pyrrolo[3,2-f]quinazolin...)
Affinity DataIC50:  300nMAssay Description:Inhibitory activity against binding to Thrombin receptor 1 (PAR-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed