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Found 1 Enz. Inhib. hit(s) with Target = 'Proteinase-activated receptor 1' and Ligand = 'BDBM50257972'
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50257972(CHEMBL4066290)
Affinity DataIC50:  3.20E+4nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed