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Found 1 Enz. Inhib. hit(s) with Target = 'Proteinase-activated receptor 1' and Ligand = 'BDBM50585042'
TargetProteinase-activated receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50585042(CHEMBL5069528)
Affinity DataIC50:  4nMAssay Description:Antagonist activity at human PAR-1 expressed in HEK293 cells assessed as reduction in TRAP induced calcium signal at 3 uM by FLIPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed