Found 2 Enz. Inhib. hit(s) with Target = 'Pyroglutamylated RF-amide peptide receptor' and Ligand = 'BDBM50020022'
Affinity DataIC50: 251nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 631nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair