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Found 3 Enz. Inhib. hit(s) with Target = 'RAC-alpha serine/threonine-protein kinase' and Ligand = 'BDBM15162'
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM15162(2-(4-{[4-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-y...)
Affinity DataIC50:  240nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt1, Akt2, and Akt3 proteins were monitored for kinase activity in the presence or absence of Akt inhibitors in a 96-well...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM15162(2-(4-{[4-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-y...)
Affinity DataIC50:  240nMAssay Description:Inhibition of Akt1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM15162(2-(4-{[4-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-y...)
Affinity DataIC50:  240nMAssay Description:Inhibition of AktMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed