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Found 4 Enz. Inhib. hit(s) with Target = 'RAC-beta serine/threonine-protein kinase' and Ligand = 'BDBM50243216'
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243216(CHEMBL443661 | N,N-dimethyl-2-(4-(6-phenyl-7-(4-((...)
Affinity DataIC50:  4nMAssay Description:Inhibition of Akt2 (unknown origin) phosphorylation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243216(CHEMBL443661 | N,N-dimethyl-2-(4-(6-phenyl-7-(4-((...)
Affinity DataIC50:  4nMAssay Description:Inhibition of Akt2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243216(CHEMBL443661 | N,N-dimethyl-2-(4-(6-phenyl-7-(4-((...)
Affinity DataIC50:  39nMAssay Description:Inhibition of Akt2 (unknown origin) by cellular assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243216(CHEMBL443661 | N,N-dimethyl-2-(4-(6-phenyl-7-(4-((...)
Affinity DataIC50:  39nMAssay Description:Inhibition of Akt2 (unknown origin) phosphorylation in human by C33a cells by IPKA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed