Found 3 Enz. Inhib. hit(s) with Target = 'Retinoic acid receptor RXR-alpha' and Ligand = 'BDBM50143827'
Affinity DataKi: 20nMAssay Description:Binding affinity for retinoid X receptor alpha (RXRalpha), using 9-cis-[3H]-retinoic acidMore data for this Ligand-Target Pair
Affinity DataEC50: 48nMAssay Description:Effective concentration for Retinoid X receptor alpha activity in CV-1 cells; Partial agonistMore data for this Ligand-Target Pair
Affinity DataEC50: 123nMAssay Description:Effective concentration for lipogenesis induced by retinoid X receptor alpha in C3H10T1/2 clone 8 fibroblast cells; Partial agonistMore data for this Ligand-Target Pair