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Found 1 Enz. Inhib. hit(s) with Target = 'Retinoic acid receptor alpha' and Ligand = 'BDBM50447837'
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
Universidade De Vigo

Curated by ChEMBL
LigandPNGBDBM50447837(CHEMBL3114297)
Affinity DataIC50:  1.28E+3nMAssay Description:Antagonist activity at Gal4-fused RARalpha (unknown origin) transfected in HEK293 cells assessed as inhibition of ATRA-induced transcriptional activi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed