TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 4.50E+3nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 1.54E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase Y181C mutant using radioactively-labeled [alpha-32P]ATP substrate and activated DNA as template-primer compl...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 1.59E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase L100I mutant using radioactively-labeled [alpha-32P]ATP substrate and activated DNA as template-primer compl...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 2.00E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase G190A mutant using radioactively-labeled [alpha-32P]ATP substrate and activated DNA as template-primer compl...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 6.33E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant using radioactively-labeled [alpha-32P]ATP substrate and activated DNA as template-primer compl...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 6.76E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase V106A mutant using radioactively-labeled [alpha-32P]ATP substrate and activated DNA as template-primer compl...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataKi: 6.99E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C mutant using radioactively-labeled [alpha-32P]ATP substrate and activated DNA as template-primer...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University
Curated by ChEMBL
Volgograd State Medical University
Curated by ChEMBL
Affinity DataIC50: 1.27E+4nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...More data for this Ligand-Target Pair