Found 4 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase MRCK gamma' and Ligand = 'BDBM2579'
TargetSerine/threonine-protein kinase MRCK gamma(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 0.190nMAssay Description:Inhibition of human DMPK2 using KKRPQRRYSNVF as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MRCK gamma(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 0.848nMAssay Description:Inhibition of human DMPK2 using KKRPQRRYSNVF as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MRCK gamma(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 37nMAssay Description:Binding constant for DMPK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase MRCK gamma(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 37nMAssay Description:Binding constant for DMPK2 kinase domainMore data for this Ligand-Target Pair