Found 9 Enz. Inhib. hit(s) with Target = 'Sodium-dependent dopamine transporter' and Ligand = 'BDBM50062915'
Affinity DataKi: 16nMAssay Description:Displacement of [3H]WIN-35,428 from human DAT expressed in mouse N2A cells after 15 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Displacement of [3H]WIN-35428 from human DAT stably expressed in mouse N2A cells by scintillation countnigMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Harvard University
Curated by PDSP Ki Database
Harvard University
Curated by PDSP Ki Database
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Harvard University
Curated by PDSP Ki Database
Harvard University
Curated by PDSP Ki Database
Affinity DataIC50: 24nMAssay Description:Inhibitory potency against [3H]DA uptake using [3H]WIN-35428 (WIN-) binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Harvard University
Curated by PDSP Ki Database
Harvard University
Curated by PDSP Ki Database
Affinity DataIC50: 83nMAssay Description:Displacement of [3H]WIN 35428 from Sprague-Dawley rat striatal tissue after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Harvard University
Curated by PDSP Ki Database
Harvard University
Curated by PDSP Ki Database
Affinity DataIC50: 83nMAssay Description:The compound was tested for its affinity at the rat striatal dopamine transporter by the displacement of [3H]WIN-35428More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Harvard University
Curated by PDSP Ki Database
Harvard University
Curated by PDSP Ki Database
Affinity DataIC50: 83nMAssay Description:Inhibitory potency against dopamine (DA) transporter using [3H]WIN-35428 (WIN-) binding assay.More data for this Ligand-Target Pair
Affinity DataIC50: 88nMAssay Description:Inhibition of [3H]-WIN- 35,428 Binding to theDopamine Transporter in Rhesus (Macaca mulatta) orCynomolgus Monkey (Macaca fascicularis) Caudate-Putame...More data for this Ligand-Target Pair
Affinity DataIC50: 156nMAssay Description:Inhibition of [3H]dopamine uptake at human DAT expressed in mouse N2A cellsMore data for this Ligand-Target Pair