Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with Target = 'Solute carrier family 15 member 1' and Ligand = 'BDBM50169127'
TargetSolute carrier family 15 member 1(Homo sapiens (Human))
Martin-Luther-University Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50169127((S)-2-((S)-2-Amino-3-carboxy-propionylamino)-succi...)
Affinity DataKi:  4.10E+5nMAssay Description:Binding affinity against membrane transport protein PEPT1 in human Caco-2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 15 member 1(Rattus norvegicus)
Kyoto University Hospital

Curated by ChEMBL
LigandPNGBDBM50169127((S)-2-((S)-2-Amino-3-carboxy-propionylamino)-succi...)
Affinity DataKi:  9.90E+5nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in PEPT1-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 15 member 1(Homo sapiens (Human))
Martin-Luther-University Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50169127((S)-2-((S)-2-Amino-3-carboxy-propionylamino)-succi...)
Affinity DataIC50:  6.30E+5nMAssay Description:Binding affinity to human PEPT1 assessed as inhibition of [14C]Gly-Sar uptake in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 15 member 1(Homo sapiens (Human))
Martin-Luther-University Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50169127((S)-2-((S)-2-Amino-3-carboxy-propionylamino)-succi...)
Affinity DataEC50:  9.90E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed