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Found 3 Enz. Inhib. hit(s) with Target = 'Solute carrier organic anion transporter family member 1A4' and Ligand = 'BDBM50375594'
TargetSolute carrier organic anion transporter family member 1A4(Rattus norvegicus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50375594(TAUROCHOLATE)
Affinity DataKi:  3.94E+4nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp2-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSolute carrier organic anion transporter family member 1A4(Rattus norvegicus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50375594(TAUROCHOLATE)
Affinity DataKi:  1.56E+5nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin uptake in Oatp2-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1A4(Rattus norvegicus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50375594(TAUROCHOLATE)
Affinity DataIC50:  1.48E+6nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In DepthDetails PubMed