Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Sphingosine 1-phosphate receptor 1' and Ligand = 'BDBM50335514'
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335514(1-((3-fluoro-4-(5-(1-phenylcyclopropyl)thiazolo[5,...)
Affinity DataEC50:  2nMAssay Description:Induction of human GFP-tagged chimeric S1P1R internalization in human U2Os cells by fluorescence microscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335514(1-((3-fluoro-4-(5-(1-phenylcyclopropyl)thiazolo[5,...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human S1P1 receptor expressed in U20S cells coexpressing eGFP assessed as receptor internalization after 1 hr by microscopy analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335514(1-((3-fluoro-4-(5-(1-phenylcyclopropyl)thiazolo[5,...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at eGFP-tagged human S1P1 receptor expressed in U2OS cells assessed as receptor internalization after 1 hr by Hoechst dye-based micr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed