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Found 5 Enz. Inhib. hit(s) with Target = 'Spindlin-1' and Ligand = 'BDBM50505574'
TargetSpindlin-1(Homo sapiens)
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50505574(CHEMBL4451634)
Affinity DataIC50:  33nMAssay Description:Displacement of trimethylated biotinylated histone H3 peptide from recombinant human His-tagged SPIN1 (26 to 262 residues) expressed in Escherichia c...More data for this Ligand-Target Pair
TargetSpindlin-1(Homo sapiens)
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50505574(CHEMBL4451634)
Affinity DataKd:  111nMAssay Description:Binding affinity to recombinant human His-tagged SPIN1 (26 to 262 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociation constan...More data for this Ligand-Target Pair
TargetSpindlin-1(Homo sapiens)
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50505574(CHEMBL4451634)
Affinity DataKd:  9.90nMAssay Description:Binding affinity to recombinant human His-tagged SPIN1 (49 to 262 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociation constan...More data for this Ligand-Target Pair
TargetSpindlin-1(Homo sapiens)
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50505574(CHEMBL4451634)
Affinity DataEC50:  270nMAssay Description:Inhibition of C-terminal Halotag-histone 3.3 tagged SPIN1 (unknown origin) transfected in human U2OS cells cotransfected with nano-luciferase at 1 uM...More data for this Ligand-Target Pair
TargetSpindlin-1(Homo sapiens)
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50505574(CHEMBL4451634)
Affinity DataKd:  55nMAssay Description:Binding affinity to human His-tagged SPIN1 (21 to 262 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant preincubat...More data for this Ligand-Target Pair