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Found 2 Enz. Inhib. hit(s) with Target = 'Steryl-sulfatase' and Ligand = 'BDBM24307'
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM24307(Letrozole derivative, 40a R-(+) | {2-bromo-4-[(R)-...)
Affinity DataIC50:  4.63E+3nMAssay Description:Inhibition of STS activity (unknown origin) expressed in JEG-3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM24307(Letrozole derivative, 40a R-(+) | {2-bromo-4-[(R)-...)
Affinity DataIC50:  4.63E+3nMAssay Description:The extent of in vitro inhibition of sulfatase activities was assessed using intact monolayers of JEG-3 cells. Sulfatase activity was measured using ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed