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Found 5 Enz. Inhib. hit(s) with Target = 'Trace amine-associated receptor 1' and Ligand = 'BDBM50336229'
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336229((+/-)-4-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-flu...)
Affinity DataKi:  4nMAssay Description:Inhibition of mouse TAAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336229((+/-)-4-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-flu...)
Affinity DataKi:  1.39E+3nMAssay Description:Inhibition of rat TAAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336229((+/-)-4-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-flu...)
Affinity DataKi: >2.00E+4nMAssay Description:Inhibition of human TAAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336229((+/-)-4-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-flu...)
Affinity DataIC50:  6nMAssay Description:Antagonist activity at mouse TAAR1 assessed as reversal of endogenous beta-PEA effectMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336229((+/-)-4-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-flu...)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human TAAR1 assessed as reversal of endogenous beta-PEA effectMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed