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Found 2 Enz. Inhib. hit(s) with Target = 'Transcription activator BRG1' and Ligand = 'BDBM646012'
TargetTranscription activator BRG1(Homo sapiens (Human))
Prelude Therapeutics

US Patent
LigandPNGBDBM646012((2S,4R)-4-hydroxy-N-[[4-(5-methyl-1,3- thiazol-4-y...)
Affinity DataIC50: <100nMAssay Description:The inhibitory activity of compounds was evaluated in vitro using TR-FRET assay with white 384-well low volume microplate (PerkinElmer ProxiPlate Plu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscription activator BRG1(Homo sapiens (Human))
Prelude Therapeutics

US Patent
LigandPNGBDBM646012((2S,4R)-4-hydroxy-N-[[4-(5-methyl-1,3- thiazol-4-y...)
Affinity DataIC50:  550nMAssay Description:The inhibitory activity of compounds was evaluated in vitro using TR-FRET assay with white 384-well low volume microplate (PerkinElmer ProxiPlate Plu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent