Found 2 Enz. Inhib. hit(s) with Target = 'Transcriptional activator protein LuxR' and Ligand = 'BDBM50265811'
TargetTranscriptional activator protein LuxR(Vibrio fischeri (strain ATCC 700601 / ES114))
University Of Wisconsin-Madison
Curated by ChEMBL
University Of Wisconsin-Madison
Curated by ChEMBL
Affinity DataIC50: 630nMAssay Description:Antagonist activity at Vibrio fischeri ES114 LuxR receptor assessed as inhibition of OHHL-induced response by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LuxR(Vibrio fischeri (strain ATCC 700601 / ES114))
University Of Wisconsin-Madison
Curated by ChEMBL
University Of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 300nMAssay Description:Agonist activity at Vibrio fischeri ES114 LuxR receptor by luciferase reporter gene assayMore data for this Ligand-Target Pair