Found 1 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily M member 8' and Ligand = 'BDBM50083037'
TargetTransient receptor potential cation channel subfamily M member 8(Rattus norvegicus (Rat))
National Research Council
Curated by ChEMBL
National Research Council
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity against rat TRPM8 expressed in HEK293 cells assessed as inhibition of icilin-induced intracellular Ca2+ level pre-treated 5 mins ...More data for this Ligand-Target Pair