Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily V member 1' and Ligand = 'BDBM50052440'
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute

Curated by ChEMBL
LigandPNGBDBM50052440(CHEMBL104647 | Phenyl-acetic acid (1aR,1bS,4aR,7aS...)
Affinity DataKi:  0.0540nMAssay Description:Inhibitory constant for RTX binding to rat spinal cordMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM50052440(CHEMBL104647 | Phenyl-acetic acid (1aR,1bS,4aR,7aS...)
Affinity DataKi:  0.120nMAssay Description:Inhibitory constant for RTX binding to porcine spinal cordMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM50052440(CHEMBL104647 | Phenyl-acetic acid (1aR,1bS,4aR,7aS...)
Affinity DataKi:  0.450nMAssay Description:Inhibitory constant for RTX binding to human spinal cordMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute

Curated by ChEMBL
LigandPNGBDBM50052440(CHEMBL104647 | Phenyl-acetic acid (1aR,1bS,4aR,7aS...)
Affinity DataKi:  600nMAssay Description:Displacement of [3H]RTX binding from Vanilloid receptor of rat dorsal Root Ganglion (DRG) membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute

Curated by ChEMBL
LigandPNGBDBM50052440(CHEMBL104647 | Phenyl-acetic acid (1aR,1bS,4aR,7aS...)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of [3H]- RTX binding to vanilloid receptor of rat urinary bladderMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM50052440(CHEMBL104647 | Phenyl-acetic acid (1aR,1bS,4aR,7aS...)
Affinity DataKi:  2.10E+3nMAssay Description:Inhibition of [3H]- RTX binding to Vanilloid receptors from pig spinal cordMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM50052440(CHEMBL104647 | Phenyl-acetic acid (1aR,1bS,4aR,7aS...)
Affinity DataKi:  6.40E+3nMAssay Description:Inhibition of [3H]- RTX binding to Vanilloid receptors from human spinal cordMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed