Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with Target = 'Type-1 angiotensin II receptor' and Ligand = 'BDBM50030690'
TargetType-1 angiotensin II receptor(RABBIT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030690(CHEMBL339113 | N-{3-[3-Butyl-4-(3-fluoro-2'-(N-t-b...)
Affinity DataIC50:  0.280nMAssay Description:In vitro inhibitory activity against Angiotensin II receptor, type 1 in rabbit aorta membrane preparations.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030690(CHEMBL339113 | N-{3-[3-Butyl-4-(3-fluoro-2'-(N-t-b...)
Affinity DataIC50:  0.280nMAssay Description:Antagonist activity at Oryctolagus cuniculus (rabbit) aortic AT1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030690(CHEMBL339113 | N-{3-[3-Butyl-4-(3-fluoro-2'-(N-t-b...)
Affinity DataIC50:  0.280nMAssay Description:In vitro inhibitory activity against Angiotensin II receptor, type 1 in rabbit aorta membrane preparations.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030690(CHEMBL339113 | N-{3-[3-Butyl-4-(3-fluoro-2'-(N-t-b...)
Affinity DataIC50:  0.281nMAssay Description:Antagonist activity at Oryctolagus cuniculus (rabbit) aortic AT1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article