Affinity DataIC50: 775nMAssay Description:Inhibition of Mer (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of tracer K5 binding to NanoLuc-fused MERTK (unknown origin) expressed in HEK293T cells measured after 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
Affinity DataKd: 570nMAssay Description:Binding affinity to human MERTK by KINOMEscan scanMAX assayMore data for this Ligand-Target Pair