Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'Vascular endothelial growth factor receptor 2' and Ligand = 'BDBM222456'
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
China Pharmaceutical University

LigandPNGBDBM222456(N-(3-fluoro-4-((2-(4-(3-(4-methylpiperazin-1-yl) p...)
Affinity DataIC50:  190nMpH: 7.4 T: 2°CAssay Description:Briefly, 20 μg/mL poly (Glu,Tyr) 4:1 (Sigma) was pre-coated in 96-well plates as a substrate. A 50 μL aliquot of 10 μmol/L ATP solutio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
China Pharmaceutical University

LigandPNGBDBM222456(N-(3-fluoro-4-((2-(4-(3-(4-methylpiperazin-1-yl) p...)
Affinity DataIC50:  190nMAssay Description:Inhibition of VEGFR-2 (unknown origin) kinase activity using poly(Glu-Tyr) at 4:1 ratio as substrate in presence of ATP incubated for 60 mins by ELIS...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
China Pharmaceutical University

LigandPNGBDBM222456(N-(3-fluoro-4-((2-(4-(3-(4-methylpiperazin-1-yl) p...)
Affinity DataIC50:  190nMAssay Description:Inhibition of VEGFR-2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed