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Found 7 Enz. Inhib. hit(s) with Target = 'Vasopressin V1a receptor' and Ligand = 'BDBM50029649'
TargetVasopressin V1a receptor(RAT)
Drugmoldesign

Curated by ChEMBL
LigandPNGBDBM50029649(1-(1-(4-(1-acetylpiperidin-4-yloxy)-2-methoxybenzo...)
Affinity DataKi:  3.70nMAssay Description:Displacement of [3H]-vasopressin from vasopressin V1a receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
Drugmoldesign

Curated by ChEMBL
LigandPNGBDBM50029649(1-(1-(4-(1-acetylpiperidin-4-yloxy)-2-methoxybenzo...)
Affinity DataKi:  3.70nMAssay Description:Binding affinity was evaluated by measuring the displacement of [3H]-AVP (arginine vasopressin) from specific binding sites in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50029649(1-(1-(4-(1-acetylpiperidin-4-yloxy)-2-methoxybenzo...)
Affinity DataKi: <2.00E+3nMAssay Description:Compound was tested for its ability to displace vasopressin from human Vasopressin V1a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50029649(1-(1-(4-(1-acetylpiperidin-4-yloxy)-2-methoxybenzo...)
Affinity DataKi:  3.20E+3nMAssay Description:Binding affinity towards human Vasopressin V1a receptor by using functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50029649(1-(1-(4-(1-acetylpiperidin-4-yloxy)-2-methoxybenzo...)
Affinity DataKi:  3.20E+3nMAssay Description:Binding affinity was evaluated by measuring the displacement of [3H]-AVP (arginine vasopressin) from specific binding sites in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50029649(1-(1-(4-(1-acetylpiperidin-4-yloxy)-2-methoxybenzo...)
Affinity DataKi:  3.20E+3nMAssay Description:Displacement of [3H]-vasopressin from vasopressin V1a receptor in human liver tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50029649(1-(1-(4-(1-acetylpiperidin-4-yloxy)-2-methoxybenzo...)
Affinity DataEC50:  3.20E+3nMAssay Description:Activity at human vasopressin V1a receptor expressed in CHO cells by NFAT-luciferase gene reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed