Affinity DataKi: >1.00E+4nMAssay Description:In vitro for histamine H1 receptor antagonist activity against histamine-induced contractions on isolated guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+4nMAssay Description:Antagonist activity at human vasopressin 1a receptor expressed in CHO cell membranes assessed as inhibition of AVP-induced IP1 accumulation by measur...More data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+4nMAssay Description:In vitro for histamine H1 receptor antagonist activity against histamine-induced contractions on isolated guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 0.158nMAssay Description:In vitro for histamine H1 receptor antagonist activity against histamine-induced contractions on isolated guinea pig ileumMore data for this Ligand-Target Pair