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Found 3 Enz. Inhib. hit(s) with Target = 'Vasopressin V1a receptor' and Ligand = 'BDBM50418365'
TargetVasopressin V1a receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418365(CHEMBL1774024)
Affinity DataKi:  0.562nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
Msd

Curated by ChEMBL
LigandPNGBDBM50418365(CHEMBL1774024)
Affinity DataKi:  4.17nMAssay Description:Displacement of [3H]AVP from rat V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Msd

Curated by ChEMBL
LigandPNGBDBM50418365(CHEMBL1774024)
Affinity DataIC50:  37.1nMAssay Description:Antagonist activity at human V1A receptor expressed in CHO cells assessed as inhibition of AVP-induced intracellular calcium releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed