Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'Vasopressin V2 receptor' and Ligand = 'BDBM301678'
TargetVasopressin V2 receptor(Homo sapiens (Human))
Ferring

US Patent
LigandPNGBDBM301678(US10131692, Compound 10)
Affinity DataEC50:  70nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetVasopressin V2 receptor(Homo sapiens (Human))
Ferring

US Patent
LigandPNGBDBM301678(US10131692, Compound 10)
Affinity DataEC50:  0.0700nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM301678(US10131692, Compound 10)
Affinity DataEC50:  0.0200nMAssay Description:Agonist activity at recombinant rat V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed