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Found 2 Enz. Inhib. hit(s) with Target = 'Vesicular acetylcholine transporter' and Ligand = 'BDBM50018079'
TargetVesicular acetylcholine transporter(Rattus norvegicus)
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50018079(5-Amino-3-(4-phenyl-piperidin-1-yl)-1,2,3,4-tetrah...)
Affinity DataKi:  40.6nMAssay Description:Displacement of (-)-[3H]vesamicol from rat VAChT expressed in rat PC12 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50018079(5-Amino-3-(4-phenyl-piperidin-1-yl)-1,2,3,4-tetrah...)
Affinity DataIC50:  100nMAssay Description:Inhibition of active transport of [3H]-Acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed