Compile Data Set for Download or QSAR
maximum 50k data
Found 83 Enz. Inhib. hit(s) with all data for entry = 50037871
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50166315(6-((3S,5S)-5-((S)-2-cyanopyrrolidine-1-carbonyl)py...)
Affinity DataIC50:  0.25nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM11113(6-{[2-({2-[(2S)-2-cyanopyrrolidin-1-yl]-2-oxoethyl...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM11056((2S)-1-[(2S)-pyrrolidin-2-ylcarbonyl]pyrrolidine-2...)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198855(3-[(2S,4S)-4-(5-methoxy-1-indolinyl)-2-pyrrolidiny...)
Affinity DataIC50:  4.80nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198844(3-{(2S,4S)-4-[N-butyl-N-(4-cyanophenylmethyl)amino...)
Affinity DataIC50:  5nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198847(3-[(2S,4S)-4-(5-fluoro-1-indolinyl)-2-pyrrolidinyl...)
Affinity DataIC50:  5.80nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198855(3-[(2S,4S)-4-(5-methoxy-1-indolinyl)-2-pyrrolidiny...)
Affinity DataIC50:  6.10nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198849(3-{(2S,4S)-4-[bis(4-cyanophenylmethyl)]amino-2-pyr...)
Affinity DataIC50:  6.40nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198875(3-[(2S,4S)-4-(5-bromo-1-indolinyl)-2-pyrrolidinylc...)
Affinity DataIC50:  6.5nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50166314(6-((3S,5S)-5-((S)-2-cyanopyrrolidine-1-carbonyl)py...)
Affinity DataIC50:  6.60nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198868(3-[(2S,4S)-4-(5-chloro-1-indolinyl)-2-pyrrolidinyl...)
Affinity DataIC50:  7nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198848(3-{(2S,4S)-4-[N-(4-cyanophenylmethyl)-N-isopropyla...)
Affinity DataIC50:  7.10nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198861(3-[(2S,4S)-4-(5-nitro-1-indolinyl)-2-pyrrolidinylc...)
Affinity DataIC50:  7.90nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198844(3-{(2S,4S)-4-[N-butyl-N-(4-cyanophenylmethyl)amino...)
Affinity DataIC50:  9.10nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198849(3-{(2S,4S)-4-[bis(4-cyanophenylmethyl)]amino-2-pyr...)
Affinity DataIC50:  9.30nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198852(3-{(2S,4S)-4-[N-(4-cyanophenylmethyl)-N-methylamin...)
Affinity DataIC50:  9.60nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198847(3-[(2S,4S)-4-(5-fluoro-1-indolinyl)-2-pyrrolidinyl...)
Affinity DataIC50:  10.1nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198861(3-[(2S,4S)-4-(5-nitro-1-indolinyl)-2-pyrrolidinylc...)
Affinity DataIC50:  10.3nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198875(3-[(2S,4S)-4-(5-bromo-1-indolinyl)-2-pyrrolidinylc...)
Affinity DataIC50:  10.7nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198841(3-[(2S,4S)-4-(1-indolinyl)-2-pyrrolidinylcarbonyl]...)
Affinity DataIC50:  11nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198848(3-{(2S,4S)-4-[N-(4-cyanophenylmethyl)-N-isopropyla...)
Affinity DataIC50:  12.5nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198868(3-[(2S,4S)-4-(5-chloro-1-indolinyl)-2-pyrrolidinyl...)
Affinity DataIC50:  13.4nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198852(3-{(2S,4S)-4-[N-(4-cyanophenylmethyl)-N-methylamin...)
Affinity DataIC50:  13.6nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198858(3-{(2S,4S)-4-[N-(4-cyanophenylmethyl)-N-(ethoxycar...)
Affinity DataIC50:  13.6nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198845(3-{(2S,4S)-4-[N-(carbamoylmethyl)-N-(4-cyanophenyl...)
Affinity DataIC50:  13.9nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198858(3-{(2S,4S)-4-[N-(4-cyanophenylmethyl)-N-(ethoxycar...)
Affinity DataIC50:  15.3nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198867(3-{(2S,4S)-4-[N-(carboxymethyl)-N-(4-cyanophenylme...)
Affinity DataIC50:  16.3nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198845(3-{(2S,4S)-4-[N-(carbamoylmethyl)-N-(4-cyanophenyl...)
Affinity DataIC50:  16.5nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198867(3-{(2S,4S)-4-[N-(carboxymethyl)-N-(4-cyanophenylme...)
Affinity DataIC50:  16.8nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198874(3-{(2S,4S)-4-[N-(4-cyanophenylmethyl)-N-(2-hydroxy...)
Affinity DataIC50:  17nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198873(((2S,4S)-4-(4-nitrophenylamino)pyrrolidin-2-yl)(th...)
Affinity DataIC50:  19.2nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198841(3-[(2S,4S)-4-(1-indolinyl)-2-pyrrolidinylcarbonyl]...)
Affinity DataIC50:  19.5nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198873(((2S,4S)-4-(4-nitrophenylamino)pyrrolidin-2-yl)(th...)
Affinity DataIC50:  21nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198874(3-{(2S,4S)-4-[N-(4-cyanophenylmethyl)-N-(2-hydroxy...)
Affinity DataIC50:  23nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198859(4-((3S,5S)-5-(thiazolidine-3-carbonyl)pyrrolidin-3...)
Affinity DataIC50:  25.2nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198863(6-((3S,5S)-5-(thiazolidine-3-carbonyl)pyrrolidin-3...)
Affinity DataIC50:  25.4nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198864(3-[(2S,4S)-4-(2-isoindolinyl)-2-pyrrolidinylcarbon...)
Affinity DataIC50:  26.4nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198859(4-((3S,5S)-5-(thiazolidine-3-carbonyl)pyrrolidin-3...)
Affinity DataIC50:  33.6nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198854(3-[(2S,4S)-4-(4-cyanophenylmethyl)amino-2-pyrrolid...)
Affinity DataIC50:  34nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198842(3-[(2S,4S)-4-(4-cyanobenzoyl)amino-2-pyrrolidinylc...)
Affinity DataIC50:  34.1nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198854(3-[(2S,4S)-4-(4-cyanophenylmethyl)amino-2-pyrrolid...)
Affinity DataIC50:  34.3nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198842(3-[(2S,4S)-4-(4-cyanobenzoyl)amino-2-pyrrolidinylc...)
Affinity DataIC50:  37.2nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198864(3-[(2S,4S)-4-(2-isoindolinyl)-2-pyrrolidinylcarbon...)
Affinity DataIC50:  39nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198853(((2S,4S)-4-(4-chlorophenylamino)pyrrolidin-2-yl)(t...)
Affinity DataIC50:  45.4nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198866(((2S,4S)-4-(4-methoxyphenylamino)pyrrolidin-2-yl)(...)
Affinity DataIC50:  51.5nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198866(((2S,4S)-4-(4-methoxyphenylamino)pyrrolidin-2-yl)(...)
Affinity DataIC50:  54.9nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198853(((2S,4S)-4-(4-chlorophenylamino)pyrrolidin-2-yl)(t...)
Affinity DataIC50:  55.1nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198871(3-{[2S,4S]-4-[3-(4-cyanophenyl)ureido]-2-pyrrolidi...)
Affinity DataIC50:  76.2nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198871(3-{[2S,4S]-4-[3-(4-cyanophenyl)ureido]-2-pyrrolidi...)
Affinity DataIC50:  85.9nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50198843(3-[(2S,4S)-4-(1,2,3,4-tetrahydro-1-quinolyl)-2-pyr...)
Affinity DataIC50:  99.8nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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